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龍圖騰網恭喜IP2IPO創新有限公司申請的專利新穎的化合物獲國家發明授權專利權，本發明授權專利權由國家知識產權局授予，授權公告號為：CN114450300B 。

龍圖騰網通過國家知識產權局官網在2025-05-20發布的發明授權授權公告中獲悉：該發明授權的專利申請號/專利號為：202080051458.3，技術領域涉及：C07K14/605；該發明授權新穎的化合物是由S·R·布魯姆設計研發完成，并于2020-06-12向國家知識產權局提交的專利申請。

本新穎的化合物在說明書摘要公布了：本發明提供了新穎的化合物，所述新穎的化合物是肽類激素類似物，并且可用于治療如糖尿病和肥胖癥等病癥。關于對胰高血糖素和GLP?1受體的效力特性，說明書中列舉的一般序列的化合物具有定制的分布。關于體內特性，已經在動物模型中證明施用本發明的示例肽會導致體重減輕增加。優選的化合物在不顯著減少食物攝入量的情況下實現這一點。

本發明授權新穎的化合物在權利要求書中公布了：1.一種式I化合物：X-W-Y1-Y2式I其中X是氨基酸序列：His1-Xaa2-Xaa3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Xaa10-Ser11-Xaa12-Xaa13-Leu14-Xaa15-Xaa16-Xaa17-Xaa18-Xaa19-Xaa20-Xaa21-Phe22-Xaa23-Xaa24-Trp25-Leu26-Xaa27-Xaa28-Xaa29-[SEQIDNO:742]W是氨基酸序列：-Xaa30-Xaa31-Xaa32-Xaa33-Xaa34-[SEQIDNO:795]；Y1是氨基酸序列：-Xaa35-Xaa36-Xaa37-Xaa38-Xaa39-Xaa40-Xaa41-Lys42-Xaa43-Xaa44[SEQIDNO:744]并且位置42的賴氨酸殘基在其ε-氨基處被Y2基團取代并且Y2是：Z-Xaa45-Xaa46-Xaa47-Xaa48-[SEQIDNO:745]并且Z為下式的基團： 其中R為C8-C28亞烷基或亞烯基，并且R1是CO2H，并且其中所述式I的化合物選自：實例號.136:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Thr47-His48-；Z＝i；R為C18直鏈亞烷基；實例號.163:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gly47-Ser48-；Z＝i；R為C16直鏈亞烷基；實例號.167:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Ser46-Gly47-Thr48-；Z＝i；R為C18直鏈亞烷基；實例號.168:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gly45-Ser46-Gly47-Ser48-；Z＝i；R為C18直鏈亞烷基；實例號.169:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Thr47-His48-；Z＝i；R為C18直鏈亞烷基；實例號.176:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gly45-Ser46-Gly47-Ser48-；Z＝i；R為C18直鏈亞烷基；實例號.195:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Ser46-Asn47-Thr48-；Z＝i；R為C18直鏈亞烷基；實例號.196:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Ser46-Gln47-Thr48-；Z＝i；R為C18直鏈亞烷基；實例號.197:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gly46-Gln47-Thr48-；Z＝i；R為C18直鏈亞烷基；實例號.198:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gln47-Thr48-；Z＝i；R為C18直鏈亞烷基；實例號.199:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Thr47-Gln48-；Z＝i；R為C18直鏈亞烷基；實例號.200:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-His47-Thr48-；Z＝i；R為C18直鏈亞烷基；實例號.201:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Asn47-His48-；Z＝i；R為C16直鏈亞烷基；實例號.202:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Thr47-His48-；Z＝i；R為C14直鏈亞烷基；實例號.203:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-His48-；Z＝i；R為C18直鏈亞烷基；實例號.204:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.205:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gln48-；Z＝i；R為C18直鏈亞烷基；實例號.211:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Ser46-Gly47-Thr48-；Z＝i；R為C18直鏈亞烷基；實例號.255:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Ser46-Gly47-Thr48-；Z＝i；R為C20直鏈亞烷基；實例號.256:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gly45-Ser46-Gly47-Ser48-；Z＝i；R為C20直鏈亞烷基；實例號.260:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Ser46-Gly47-Thr48-；Z＝i；R為C22直鏈亞烷基；實例號.261:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gly45-Ser46-Gly47-Ser48-；Z＝i；R為C22直鏈亞烷基；實例號.262:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.263:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gln48-；Z＝i；R為C18直鏈亞烷基；實例號.264:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Asn48-；Z＝i；R為C20直鏈亞烷基；實例號.265:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gln48-；Z＝i；R為C20直鏈亞烷基；實例號.266:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-Gln48-；Z＝i；R為C18直鏈亞烷基；實例號.267:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Lys42；Y2＝Z-Gln48-；Z＝i；R為C18直鏈亞烷基；實例號.268:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Gly39-Lys42；Y2＝Z-Gln48-；Z＝i；R為C18直鏈亞烷基；實例號.269:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gln48-；Z＝i；R為C18直鏈亞烷基；實例號.270:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gln47-Gly48-；Z＝i；R為C18直鏈亞烷基；實例號.271:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gly47-Gln48-；Z＝i；R為C18直鏈亞烷基；實例號.272:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gly47-Gln48-；Z＝i；R為C22直鏈亞烷基；實例號.273:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Ser46-Gly47-Thr48-；Z＝i；R為C18直鏈亞烷基；實例號.276:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gln48-；Z＝i；R為C18直鏈亞烷基；實例號.277:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Ser46-Gly47-Thr48-；Z＝i；R為C18直鏈亞烷基；實例號.278:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gln48-；Z＝i；R為C16直鏈亞烷基；實例號.289:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Ser46-Gly47-Thr48-；Z＝i；R為C16直鏈亞烷基；實例號.290:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gly47-Ser48-；Z＝i；R為C16直鏈亞烷基；實例號.301:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Asn47-His48-；Z＝i；R為C16直鏈亞烷基；實例號.314:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Asn47-His48-；Z＝i；R為C18直鏈亞烷基；實例號.315:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-Asn47-His48-；Z＝i；R為C16直鏈亞烷基；實例號.316:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gln47-His48-；Z＝i；R為C16直鏈亞烷基；實例號.317:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-Asn47-His48-；Z＝i；R為C16直鏈亞烷基；實例號.319:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-Asn47-His48-；Z＝i；R為C16直鏈亞烷基；實例號.321:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Asn47-His48-；Z＝i；R為C16直鏈亞烷基；實例號.323:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Asn47-His48-；Z＝i；R為C16直鏈亞烷基；實例號.325:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.327:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.329:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Asn48-；Z＝i；R為C16直鏈亞烷基；實例號.340:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Ser46-Gly47-Thr48-；Z＝i；R為C14直鏈亞烷基；實例號.341:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-His32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Gly47-Ser48-；Z＝i；R為C14直鏈亞烷基；實例號.366:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-Gly47-Ser48-；Z＝i；R為C16直鏈亞烷基；實例號.367:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-Thr45-Gly46-Ser47-Gly48-；Z＝i；R為C16直鏈亞烷基；實例號.368:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-Asn48-；Z＝i；R為C16直鏈亞烷基；實例號.369:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-Gln48-；Z＝i；R為C16直鏈亞烷基；實例號.412:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-Thr45-Gly46-Ser47-Gly48-；Z＝i；R為C18直鏈亞烷基；實例號.521:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-His32-Pro33-Ser34-Pro35-Pro36-Pro37-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.536:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.537:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.538:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.542:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-Gln30-Gln31-His32-Glu33-Ser34-Pro35-Pro36-Pro37-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.543:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-Gln30-Gln31-His32-Glu33-Ser34-Pro35-Pro36-Pro37-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.544:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-His32-Pro33-Ser34-Pro35-Pro36-Pro37-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.549:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-Gln33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.550:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-Gln33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.552:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-His32-Gln33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.553:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-Gln33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.581:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-Pro33-Ser34-Pro35-Pro36-Pro37-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.588:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-His20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-Glu34-Ser35-Pro36-Pro37-Pro38-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.589:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-His20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-Ser34-Pro35-Pro36-Pro37-Lys42；Y2＝Z-Gly47-Ser48-；Z＝i；R為C18直鏈亞烷基；實例號.590:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-His20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-Ser34-Pro35-Pro36-Pro37-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.595:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-His32-Glu33-Ser34-Pro35-Pro36-Pro37-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.597:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-His32-Glu33-Ser34-Pro35-Pro36-Pro37-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.598:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-Glu34-Ser35-Pro36-Pro37-Pro38-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.602:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-Gln33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.603:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.604:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-Glu34-Ser35-Pro36-Pro37-Pro38-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.605:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-His20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.606:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-His20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-His32-Glu33-Ser34-Pro35-Pro36-Pro37-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.632:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-His32-Gln33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.636:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-His32-Gln33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.638:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-His32-Gln33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.639:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-His32-Gln33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.642:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.643:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.646:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-Gln33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.647:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-Gln33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.652:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-His20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-Glu34-Ser35-Pro36-Pro37-Pro38-Gly39-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.653:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-His20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-Glu34-Ser35-Pro36-Pro37-Pro38-Gly39-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.654:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.655:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-Ser34-Glu35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.656:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.657:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-Gln30-His31-Gln32-His33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.658:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-Gln30-Gln31-His32-Glu33-Ser34-Glu35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.660:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-Gln33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.661:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-Gln33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.663:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-Gln30-Gln31-His32-Glu33-Ser34-Pro35-Pro36-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.671:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-Gln30-Gln31-His32-Glu33-Ser34-Ser35-Gly36-Ala37-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.672:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-His32-Glu33-Ser34-Ser35-Gly36-Ala37-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.673:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-His20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-Glu34-Ser35-Ser36-Ala37-Ser38-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.678:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-Gln30-Gln31-His32-Glu33-Ser34-Ser35-Gly36-Ala37-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.682:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-Gln33-His34-Glu35-Gly36-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.691:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-Gln33-His34-Glu35-Ser36-Pro37-Pro38-Gly39-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.695:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-Gln33-His34-Glu35-Ser36-Ser37-Ser38-Gly39-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.700:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-His20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-Glu34-Ser35-Pro36-Pro37-Pro38-Gly39-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.701:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-Gln33-His34-Glu35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.704:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Arg20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-Glu34-Ser35-Pro36-Pro37-Pro38-Gly39-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.705:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Arg20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-Pro34-Ser35-Pro36-Pro37-Pro38-Gly39-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.706:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-Pro34-Ser35-Pro36-Pro37-Pro38-Gly39-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.707:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-Pro34-Ser35-Ser36-Ser37-Ser38-Ala39-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.708:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-Pro34-Ser35-Ser36-Ser37-Ala38-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.709:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-His20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-Pro34-Ser35-Ser36-Ser37-Ala38-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；實例號.711:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-His34-Pro35-Ser36-Ser37-Ser38-Ala39-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.712:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-His31-Gln32-Gln33-His34-Pro35-Ser36-Pro37-Pro38-Pro39-Gly40-Lys42；Y2＝Z-；Z＝i；R為C18直鏈亞烷基；實例號.725:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Gln20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-Pro34-Ser35-Ser36-Ser37-Ala38-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基；并且實例號.726:His1-AIB2-His3-Gly4-Thr5-Phe6-Thr7-Ser8-Asp9-Tyr10-Ser11-Lys12-Tyr13-Leu14-Asp15-Ala16-Lys17-Arg18-Ala19-Arg20-Glu21-Phe22-Ile23-Glu24-Trp25-Leu26-Leu27-Gln28-Ser29-His30-Gln31-Gln32-His33-Pro34-Ser35-Ser36-Ser37-Ala38-Lys42；Y2＝Z-Asn48-；Z＝i；R為C18直鏈亞烷基。

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